Articles
Reports
Articles
Gomes RFA, Ravasco JMJM, Andrade KHS, Coelho JAS, Moreira R, Oliveira R, Nogueira F, Afonso CAM. Tandem Thio-Michael Addition/Remote Lactone Activation of 5-Hydroxymethylfurfural-Derived δ-Lactone-Fused Cyclopentenones. ChemSusChem. 2022; e202102204. DOI: 10.1002/cssc.202102204.
- April 27, 2022
- Bioorganic Chemistry
Vale FF, Vítor J, Marques AT, Azevedo-Pereira JM, Anes E, Goncalves J. Origin, phylogeny, variability and epitope conservation of SARS-CoV-2 worldwide. Virus Res. 2021; 304, 198526. DOI: 10.1016/j.virusres.2021.198526.
- October 15, 2021
- Molecular Microbiology and Biotechnology
Fernandez-Checa JC, Bagnaninchi P, Ye H, Sancho-Bru P, Falcon-Perez JM, Royo F, Garcia-Ruiz C, Konu O, Miranda J, Lunov O, Dejneka A, Elfick A, McDonald A, Sullivan GJ, Aithal GP, Lucena MI, Andrade RJ, Fromenty B, Kranendonk M, Cubero FJ, Nelson LJ. Advanced preclinical models for evaluation of drug-induced liver injury – consensus statement by the European Drug-Induced Liver Injury Network [PRO-EURO-DILI-NET]. J Hepatol. 2021; 75 (4): 935-959. DOI: 10.1016/j.jhep.2021.06.021
Lee K, Yang A, Lin Y-C, Reker D, Bernardes G.J.L., Rodrigues T. Combating small molecule aggragation with machine learning. Cell Reports Physical Science 2021; 2 (9): 100573. DOI: 10.1016/j.xcrp.2021.100573
- September 22, 2021
- Medicinal Chemistry
Valente E, Testa B, Constantino L. Activation of benzoate model prodrugs by mycobacteria. Comparison with mammalian plasma and liver hydrolysis. Eur J Pharm Sci. 2021, 162:105831. DOI: 10.1016/j.ejps.2021.105831.
- July 1, 2021
- Medicinal Organic Chemistry
Gomes-Alves AG, Duarte M, Cruz T, Castro H, Lopes F, Moreira R, Ressurreição AS, Tomás AM. Quinolin-(1H)-imines as a new chemotype against leishmaniasis: biological evaluation and mechanistic studies. Antimicrob Agents Chemother 2021; Apr 26:AAC.01513-20. DOI: 10.1128/AAC.01513-20.
- June 17, 2021
- Medicinal Chemistry
Cardoso R; Guo F; Heisser T; Hackl M; Ihle P; De Schutter H; Van Damme N; Valerianova Z; Atanasov T; Májek O; Mužík J; Nilbert MC; Tybjerg AJ; Innos K; Mägi M; Malila N; Bouvier A-M; Bouvier V; Launoy G; Woronoff A-S; Cariou M; Robaszkiewicz M; Delafosse P; Poncet F; Katalinic A; Walsh PM; Senore C; Rosso S; Vincerževskienė I; Lemmens V.E.P.P.; Elferink M.A.G.; Johannesen TB; Kørner H; Pfeffer F; Bento MJ; Rodrigues J; Alves da Costa F; Miranda A; Zadnik V; Žagar T; Marques A.L.M.; Marcos-Gragera R; Puigdemont M; Galceran J; Carulla M; Chirlaque M-D; Ballesta M; Sundquist K; Sundquist J; Weber M; Jordan A; Herrmann C; Mousavi M; Ryzhov A; Hoffmeister M; Brenner H. Colorectal cancer incidence, mortality, and stage distribution in European countries in the colorectal cancer screening era: an international population-based study. The Lancet Oncology. 2021; 22 (7): 1002-1013. DOI: 10.1016/S1470-2045(21)00199-6
- May 25, 2021
- Pharmaceutical Care and Clinical Pharmacy
Figueira I, Godinho-Pereira J, Galego S, Maia J, Haskó J, Molnár K, Malhó R, Costa-Silva B, Wilhelm I, Krizbai IA, Brito MA. MicroRNAs and extracellular vesicles as distinctive biomarkers of precocious and advanced stages of breast cancer brain metastases development. Int J Mol Sci 2021; 22: 5214. DOI: 10.3390/ijms22105214
- May 14, 2021
- Neurovascular
Carreira AC, Pokorna S, Ventura AE, Walker MW, Futerman, AH, Lloyd-Evans E, de Almeida RFM, Silva LC. Biophysical impact of sphingosine and other abnormal lipid accumulation in Niemann-Pick disease type C cell models. Biochim Biophys Acta Mol Cell Biol Lipids. 2021; 1866: 158944. DOI: 10.1016/j.bbalip.2021.158944.
- May 1, 2021
- Drug Delivery & Immunoengineering
Raimundo L, Paterna A, Calheiros J, Ribeiro J, Cardoso DSP, Piga I, Neto SJ, Hegan D, Glazer PM, Indraccolo S, Mulhovo S, Costa JL, Ferreira MJU, Saraiva S. BBIT20 inhibits homologous DNA repair with disruption of the BRCA1–BARD1 interaction in breast and ovarian cancer. Br J Pharmacol 2021, 3627–3647, DOI:10.1111/bph.15506.
- April 26, 2021
- Natural Products Chemistry
Reports